Hormone antagonists / / ed. by M.K. Agarwal.

• Superior document: Title is part of eBook package: De Gruyter DGBA Medicine and Life Sciences - <1990
• MitwirkendeR: Abe, Youichi,; Agarwal, M. K.,; Andries, Maria,; Baillet, Jack,; Bell, Philip A.,; Benco, Rosanna,; Bex, Frederick,; Black, Larry J.,; Blake, Colin C.P.,; Burridge, Jane M.,; Cake, Max H.,; Catt, Kevin J.,; Clark, James H.,; Corbin, Alan,; Daniel, Paul,; Davies, Peter,; Denef, Cali,; Dry, J.,; Duax, William L.,; Evans, Rawden W.,; Fabre-Nys, Claude,; Ferrari, Carlo,; Friesen, H.G.,; Gardner, Jerry D.,; Gless, Kurt-Holger,; Gold, Mark S.,; Griffin, Jane F.,; Guthrie, Sylvia C.,; Haack, Doris,; Hampl, Richard,; Harwood, James P.,; Helber, Albert,; Hendry, William J.,; Hiraga, Kentaro,; Hirst, Barry H.,; Ho, Kevin K.W.,; Hruby, Victor J.,; Inaba, N.,; Jensen, Robert T.,; Jones, T. Ryland,; Jordan, V. Craig,; Kassen, Nadim,; Keene, Jeffery L.,; Kendle, K.E.,; Komori, Tadamitsu,; Leavitt, Wendell W.,; Limbird, Lee E.,; Maeda, Yoshiaki,; Markavarich, Barry M.,; McCormack, Shirley A.,; McDonald, Richard G.,; Miki, Takuichi,; Miura, Katsuyuki,; Mosberg, Henry I.,; Murphy, Leigh C.,; Nakayama, Ryo,; Naylor, Paul H.,; Neri, Rudolph,; Nicholson, Robert I.,; Nishizawa, Yasuko,; Noma, Keizo,; Oatley, Stuart J.,; Okulicz, William C.,; Paillard, Jacques,; Pottash, A. Carter,; Pradalier, A.,; Rampini, Pietro,; Ramsay, Lawrence E.,; Robidoux, William F.,; Rohrer, Douglas C.,; Rosen, Fred,; Ross, Patrick,; Ruh, Thomas S.,; Sato, Bunzo,; Sekiya, S.,; Sonino, Nicoletta,; Starka, Lubos,; Sutherland, Robert L.,; Syne, Joy S.,; Takamizawa, H.,; Vecsei, Paul,; Vickery, Brian H.,; Wambach, Gerhard,; Waters, M.J.,; Watta, Colin K.W.,; Weeks, Charles M.,; Yamamoto, Kenjiro,; Yamamura, Matsumoto,; Yamamura, Yuichi,; Yeoh, George C.T.,; Yoshimoto, Shinobu,
• HerausgeberIn: Agarwal, M.K.,
• Place / Publishing House: Berlin ;, Boston : : De Gruyter, , [2019]; ©1982
• Year of Publication: 2019
• Edition: Reprint 2019
• Language: English
• Physical Description: 1 online resource (IX, 732 p.) :; Num. figs.

Table of Contents

Frontmatter -- PREFACE -- CONTENTS -- SECTION 1: STEROID HORMONE ANTAGONISTS -- STEROID AGONISTS AND ANTAGONISTS: MOLECULAR CONFORMATION, RECEPTOR BINDING AND ACTIVITY -- ANTIHORMONAL ACTIVITIES OF STEROIDS WITH MODIFIED RINGS A OR B -- ANTAGONISM OF STEROID HORMONES BY SPECIFIC ANTIBODIES -- ANTAGONISM OF STEROID HORMONE ACTION BY INTERFERENCE OF RECEPTOR FUNCTION WITH LOW MOLECULAR WEIGHT INHIBITORS -- ANTI-STEROIDS AND ANIMAL BEHAVIOUR : A REVIEW -- AGONISTIC AND ANTAGONISTIC PROPERTIES OF CLOMIPHENE -- HYDROXYLATED ANTIOESTROGENS: NEW PHARMACOLOGICAL PROBES TO INVESTIGATE OESTROGEN AND ANTIOESTROGEN ACTION -- Biological Actions and Binding Properties of a New Estrogen Antagonist -- BINDING PROPERTIES AND LIGAND SPECIFICITY OF AN INTRACELLULAR BINDING SITE WITH SPECIFICITY FOR SYNTHETIC OESTROGEN ANTAGONISTS OF THE TRIPHENYLETHYLENE SERIES -- ESTROGEN RECEPTOR BINDING PARAMETERS OF THE HIGH AFFINITY ANTIESTROGEN 3H-H1285 -- POTENTIAL ANTIOESTROGENIC AND ANTITUMOUR MECHANISMS OF TAMOXIFEN ACTION IN BREAST CANCER -- ANTI-TUMOR ACTION OF NON-STEROIDAL ANTIESTROGENS -- PROGESTERONE INHIBITION OF NUCLEAR ESTROGEN RECEPTOR RETENTION -- ADVANCES IN THE STUDY OF ANTIPROGESTATIONAL AGENTS -- PHARMACOLOGICAL AND CLINICAL EFFECTS OF ANT IANDROGENS -- MECHANISM OF ACTION OF A STEROIDAL ANTI-ANDROGEN TSAA-291, 16B-ETHYL-176-H YDROXYESTR-4-EN-3-ONE -- STRUCTURE-AFFINITY RELATIONSHIP OF ANTIMINERALOCORTICOID ACTIVE STEROIDS -- PROGESTIN ANTAGONISM OF ALDOSTERONE ACTION IN THE KIDNEY -- CLINICAL PHARMACOLOGY AND THERAPEUTIC USE OF ALDOSTERONE ANTAGONISTS -- ANTIGLUCOCORTICOIDS: DIFFERENTIAL ANTAGONISM OF IN VIVO RESPONSES TO DEXAMETHASONE -- ANTAGONISM OF GLUCOCORTICOID ACTION IN VIVO -- DISCRIMINATION BETWEEN GLUCOCORTICOID AGONISTS AND ANTAGONISTS BY MEANS OF RECEPTOR BINDING STUDIES -- ANTAGONISM OF GLUCOCORTICOID ACTION BY INSULIN -- INHIBITION OF ADRENAL STEROID BIOSYNTHESIS BY METYRAPONE -- SECTION 2: PEPTIDE HORMONE ANTAGONISTS -- STRUCTURAL, CONFORMATIONAL AND DYNAMIC CONSIDERATIONS IN THE DEVELOPMENT OF PEPTIDE HORMONE ANTAGONISTS -- INHIBITORS OF THE RENIN-ANGIOTENSIN SYSTEM -- ANTI-PROLACTIN AND ANTI-GROWTH HORMONE RECEPTOR ANTIBODIES, AND THEIR USE AS ANTI-HORMONAL AGENTS -- CLINICAL APPLICATIONS OF PROLACTIN LOWERING DRUGS -- RECEPTOR ANTAGONISTS OF THE ACTIONS OF GASTROINTESTINAL PEPTIDES ON PANCREATIC ACINAR CELLS -- GASTHIN ANTAGONISM -- ANTIGONADAL EFFECTS OF GONADOTROPIN-RELEASING HORMONE AND AGONIST ANALOGS -- ANTAGONISTS OF HYPOTHALAMIC REGULATORY PEPTIDES AND DOPAMINE -- LUTEINIZING HORMONE RELEASING HORMONE ANALOGS AS ANTIHORMONES -- ANTIGONADOTROPIC, ANTISTEROIDOGENIC AND ANTISTEROIDAL ACTIVITIES OF AGONIST ANALOGS OF LUTEINIZING HORMONERELEASING HORMONE AS REVEALED BY THEIR ANTIREPRODUCTIVE ACTIVITIES -- SECTION 3: MISCELLANEOUS HORMONES AND ANTAGONISTS -- HORMONAL INHIBITION OF ADENYLATE CYCLASE: A POSSIBLE MECHANISM FOR PHYSIOLOGICAL ANTAGONISM -- NALOXONE AND NALTREXONE: Endorphin Antihormones -- ANTIHISTAMINES -- X-RAY CRYSTALLOGRAPHIC STUDIES OF THYROID HORMONE, ANALOGUE AND COMPETITOR BINDING INTERACTIONS WITH HUMAN SERUM PREALBUMIN -- ANTIPHEROMONES? -- AUTHOR INDEX -- SUBJECT INDEX -- Backmatter