Hormone antagonists / / ed. by M.K. Agarwal.
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Other title: | Frontmatter -- PREFACE -- CONTENTS -- SECTION 1: STEROID HORMONE ANTAGONISTS -- STEROID AGONISTS AND ANTAGONISTS: MOLECULAR CONFORMATION, RECEPTOR BINDING AND ACTIVITY -- ANTIHORMONAL ACTIVITIES OF STEROIDS WITH MODIFIED RINGS A OR B -- ANTAGONISM OF STEROID HORMONES BY SPECIFIC ANTIBODIES -- ANTAGONISM OF STEROID HORMONE ACTION BY INTERFERENCE OF RECEPTOR FUNCTION WITH LOW MOLECULAR WEIGHT INHIBITORS -- ANTI-STEROIDS AND ANIMAL BEHAVIOUR : A REVIEW -- AGONISTIC AND ANTAGONISTIC PROPERTIES OF CLOMIPHENE -- HYDROXYLATED ANTIOESTROGENS: NEW PHARMACOLOGICAL PROBES TO INVESTIGATE OESTROGEN AND ANTIOESTROGEN ACTION -- Biological Actions and Binding Properties of a New Estrogen Antagonist -- BINDING PROPERTIES AND LIGAND SPECIFICITY OF AN INTRACELLULAR BINDING SITE WITH SPECIFICITY FOR SYNTHETIC OESTROGEN ANTAGONISTS OF THE TRIPHENYLETHYLENE SERIES -- ESTROGEN RECEPTOR BINDING PARAMETERS OF THE HIGH AFFINITY ANTIESTROGEN 3H-H1285 -- POTENTIAL ANTIOESTROGENIC AND ANTITUMOUR MECHANISMS OF TAMOXIFEN ACTION IN BREAST CANCER -- ANTI-TUMOR ACTION OF NON-STEROIDAL ANTIESTROGENS -- PROGESTERONE INHIBITION OF NUCLEAR ESTROGEN RECEPTOR RETENTION -- ADVANCES IN THE STUDY OF ANTIPROGESTATIONAL AGENTS -- PHARMACOLOGICAL AND CLINICAL EFFECTS OF ANT IANDROGENS -- MECHANISM OF ACTION OF A STEROIDAL ANTI-ANDROGEN TSAA-291, 16B-ETHYL-176-H YDROXYESTR-4-EN-3-ONE -- STRUCTURE-AFFINITY RELATIONSHIP OF ANTIMINERALOCORTICOID ACTIVE STEROIDS -- PROGESTIN ANTAGONISM OF ALDOSTERONE ACTION IN THE KIDNEY -- CLINICAL PHARMACOLOGY AND THERAPEUTIC USE OF ALDOSTERONE ANTAGONISTS -- ANTIGLUCOCORTICOIDS: DIFFERENTIAL ANTAGONISM OF IN VIVO RESPONSES TO DEXAMETHASONE -- ANTAGONISM OF GLUCOCORTICOID ACTION IN VIVO -- DISCRIMINATION BETWEEN GLUCOCORTICOID AGONISTS AND ANTAGONISTS BY MEANS OF RECEPTOR BINDING STUDIES -- ANTAGONISM OF GLUCOCORTICOID ACTION BY INSULIN -- INHIBITION OF ADRENAL STEROID BIOSYNTHESIS BY METYRAPONE -- SECTION 2: PEPTIDE HORMONE ANTAGONISTS -- STRUCTURAL, CONFORMATIONAL AND DYNAMIC CONSIDERATIONS IN THE DEVELOPMENT OF PEPTIDE HORMONE ANTAGONISTS -- INHIBITORS OF THE RENIN-ANGIOTENSIN SYSTEM -- ANTI-PROLACTIN AND ANTI-GROWTH HORMONE RECEPTOR ANTIBODIES, AND THEIR USE AS ANTI-HORMONAL AGENTS -- CLINICAL APPLICATIONS OF PROLACTIN LOWERING DRUGS -- RECEPTOR ANTAGONISTS OF THE ACTIONS OF GASTROINTESTINAL PEPTIDES ON PANCREATIC ACINAR CELLS -- GASTHIN ANTAGONISM -- ANTIGONADAL EFFECTS OF GONADOTROPIN-RELEASING HORMONE AND AGONIST ANALOGS -- ANTAGONISTS OF HYPOTHALAMIC REGULATORY PEPTIDES AND DOPAMINE -- LUTEINIZING HORMONE RELEASING HORMONE ANALOGS AS ANTIHORMONES -- ANTIGONADOTROPIC, ANTISTEROIDOGENIC AND ANTISTEROIDAL ACTIVITIES OF AGONIST ANALOGS OF LUTEINIZING HORMONERELEASING HORMONE AS REVEALED BY THEIR ANTIREPRODUCTIVE ACTIVITIES -- SECTION 3: MISCELLANEOUS HORMONES AND ANTAGONISTS -- HORMONAL INHIBITION OF ADENYLATE CYCLASE: A POSSIBLE MECHANISM FOR PHYSIOLOGICAL ANTAGONISM -- NALOXONE AND NALTREXONE: Endorphin Antihormones -- ANTIHISTAMINES -- X-RAY CRYSTALLOGRAPHIC STUDIES OF THYROID HORMONE, ANALOGUE AND COMPETITOR BINDING INTERACTIONS WITH HUMAN SERUM PREALBUMIN -- ANTIPHEROMONES? -- AUTHOR INDEX -- SUBJECT INDEX -- Backmatter |
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Format: | Mode of access: Internet via World Wide Web. |
ISBN: | 9783111506753 9783110637861 |
DOI: | 10.1515/9783111506753 |
Access: | restricted access |
Hierarchical level: | Monograph |
Statement of Responsibility: | ed. by M.K. Agarwal. |
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