Enzyme Inhibitor from Marine Organisms

Marine habitats are promising sources to identify novel organisms and compounds. A total of 70% of the planet’s surface is covered by ocean, and little is known about the biosphere within these habitats. In the last few years, numerous novel bioactive compounds or secondary metabolites from marine e...

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Year of Publication:2020
Language:English
Physical Description:1 electronic resource (130 p.)
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(oapen)https://directory.doabooks.org/handle/20.500.12854/69424
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spelling Tischler, Dirk edt
Enzyme Inhibitor from Marine Organisms
Basel, Switzerland MDPI - Multidisciplinary Digital Publishing Institute 2020
1 electronic resource (130 p.)
text txt rdacontent
computer c rdamedia
online resource cr rdacarrier
Marine habitats are promising sources to identify novel organisms and compounds. A total of 70% of the planet’s surface is covered by ocean, and little is known about the biosphere within these habitats. In the last few years, numerous novel bioactive compounds or secondary metabolites from marine environments have been described. This is, and will be, a promising source of candidate compounds in pharma research and chemical biology. In recent years, a number of novel techniques have been introduced to the field and it has become easier to actually (bio-)prospect compounds such as enzyme inhibitors. Those novel compounds then need to be characterized and evaluated in comparison to well-known representatives. This Special Issue focuses on the description of novel enzyme inhibitors of marine origin, including bioprospecting, omic approaches, and structural and mechanistic aspects.
English
Research & information: general bicssc
sponge Monanchora pulchra
pentacyclic guanidine alkaloids
GH36 α-galactosidase
GH109 α-N-acetylgalactosaminidase
slow-binding irreversible inhibitor
monanchomycalin B
monanhocidin A
normonanhocidin A
Alzheimer′s disease
BACE1
acetylcholinesterase
in silico docking
phlorotannins
Ulva intestinalis
ACE inhibitory peptide
optimization
purification
structural identification
molecular docking
secondary metabolites
Mycosphaerella sp.
asperchalasine
α-glucosidase
kinase inhibitors
drug development
marine natural products
inhibitor
macroalgae
marine fish
protease
Ulva ohnoi
functional annotation
structure–function relation
natural products
bioactives
enzyme inhibition
inactivation
marine bacteria
marine fungi
marine sponges
3-03943-783-6
3-03943-784-4
Tischler, Dirk oth
language English
format eBook
author2 Tischler, Dirk
author_facet Tischler, Dirk
author2_variant d t dt
author2_role Sonstige
title Enzyme Inhibitor from Marine Organisms
spellingShingle Enzyme Inhibitor from Marine Organisms
title_full Enzyme Inhibitor from Marine Organisms
title_fullStr Enzyme Inhibitor from Marine Organisms
title_full_unstemmed Enzyme Inhibitor from Marine Organisms
title_auth Enzyme Inhibitor from Marine Organisms
title_new Enzyme Inhibitor from Marine Organisms
title_sort enzyme inhibitor from marine organisms
publisher MDPI - Multidisciplinary Digital Publishing Institute
publishDate 2020
physical 1 electronic resource (130 p.)
isbn 3-03943-783-6
3-03943-784-4
illustrated Not Illustrated
work_keys_str_mv AT tischlerdirk enzymeinhibitorfrommarineorganisms
status_str n
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carrierType_str_mv cr
is_hierarchy_title Enzyme Inhibitor from Marine Organisms
author2_original_writing_str_mv noLinkedField
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